Andrew Leach

Andrew Leach

Dr

  • Lecturer in Pharmaceutical Chemistry, Pharmacy
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  • 2011

    4- (PYRIMIDIN-2-YL) -PIPERAZINE AND 4- (PYRIMIDIN-2-YL) -PIPERIDINE DERIVATIVES AS GPR119 MODULATORS

    Birch, Alan, M., Broo, Dan, A., Butlin, Roger, J., Scott, James, S., Clarke, David, S., Davidsson, Ojvind, P., De La Motte, H., Johansson, Kjell, E., Leach, A., MacFaul, Philip, A., O'Donnell, Charles, J. & Whittamore, Paul, Robert, O., 17 Mar 2011, IPC No. C07D 413/ 14 A I, Patent No. WO2011030139, Priority date 15 Feb 2010, Priority No. US20100304564P

    Research output: Patent

  • 4 -AMINO -7,8- DIHYDROPYRIMIDO [5, 4 - F] [1, 4] OXAZEPIN- 5 ( 6H) - ONE BASED DGAT1 INHIBITORS

    Birch, Alan, M., Goldberg, Frederick, W. & Leach, A., 6 Oct 2011, IPC No. A61P 3/ 10 A I, Patent No. WO2011121350, Priority date 27 Jul 2010, Priority No. US20100368040P

    Research output: Patent

  • Adamantyl Iminocarbonyl-Substituted Pyrimidines As Inhibitors Of 11-Beta-HSD1 826

    Bennett Stuart Norman, L., Goldberg Frederick, W., Leach, A., Whittamore Paul Robert, O. & Soerme, P., 21 Apr 2011, IPC No. C07D 239/ 47 A I, Patent No. US2011092526, Priority date 19 Oct 2010, Priority No. US20100907056

    Research output: Patent

  • Therapeutic agents

    Johansson, K. E., Birch, A. M., De La Motte, H., Butlin, R. J., Clarke, D. S., Leach, A., MacFaul, P. A., O'Donnell, C. J., Scott, J. S., Whittamore, P. R. O., Broo, D. A. & Davidsson, O. P., 1 May 2011, IPC No. A61P 3/ 10 A N, Patent No. TW201114759, Priority date 15 Feb 2010, Priority No. US20100304564P

    Research output: Patent

  • Therapeutic Agents 812

    Johansson Kjell, E., Birch Alan, M., De La Motte, H., Butlin Roger, J., Clarke David, S., Leach, A., MacFaul Philip, A., O'Donnell Charles, J., Scott James, S., Whittamore Paul Robert, O., Broo Dan, A. & Davidsson Oejvind, P., 17 Mar 2011, IPC No. C07D 487/ 08 A I, Patent No. US2011065706, Priority date 10 Sep 2010, Priority No. US20100879631

    Research output: Patent

  • 2010

    PYRAZINE CARBOXAMIDES AS INHIBITORS OF DGAT1

    Birch, A. M., Butlin, R. J., Campbell, L., Green, C., Leach, A., Murray, P. M., Ryberg, P. O. & Waring, M. J., 23 Dec 2010, IPC No. C07D 413/ 10 A I, Patent No. WO2010146395, Priority date 19 Jun 2009, Priority No. US20090218539P

    Research output: Patent

  • 2009

    CARBAMOYL COMPOUNDS AS DGAT1 INHIBITORS 190

    Petersson, Annika, U., Bauer, Udo, A., Birch, Alan, M., Butlin, Roger, J., Green, C., Barlind, Jonas, G., Hovland, R., Johannesson, P., Johansson, Jan, M., Leach, A. & Noeske, Alexander, T., 2 Jul 2009, IPC No. C07D 403/ 10 A I, Patent No. WO2009081195, Priority date 20 Dec 2007, Priority No. US20070015397P

    Research output: Patent

  • SUBSTITUTED PYRIMIDIN-5-CARBOXAMIDES 281

    Gill, Adrian, L., Leach, A., Packer, M., Scott, James, S., Soerme, P., Swales, John, G. & Whittamore, Paul, Robert, O., 29 Oct 2009, IPC No. C07D 417/ 04 A I, Patent No. WO2009130496, Priority date 23 Dec 2008, Priority No. US20080140201P

    Research output: Patent

  • 2008

    PIPERIDINE DERIVATIVES FOR THE TREATMENT OF OBESITY

    Butlin, Roger, J., Caulkett, Peter, William, R., Leach, A., Newcombe, Nicholas, J., O'Donnell, Charles, J. & Wood, James, M., 26 Jun 2008, IPC No. C07D 473/ 34 A I, Patent No. WO2008075064, Priority date 5 Apr 2007, Priority No. US20070910268P

    Research output: Patent

  • PIPERIDINE DERIVATIVES FOR THE TREATMENT OF OBESITY

    Butlin, Roger, J., Caulkett, Peter, William, R., Leach, A., Newcombe, Nicholas, J., O'Donnell, Charles, J. & Wood, James, M., 26 Jun 2008, IPC No. C07D 401/ 12 A I, Patent No. WO2008075077, Priority date 29 Mar 2007, Priority No. US20070908706P

    Research output: Patent

  • SUBSTITUTED PIPERIDINES HAVING PROTEIN KINASE INHIBITING ACTIVITY

    Caldwell, J., Da Fonseca McHardy, Tatiana, F., Luke, Richard, William, A., Matusiak, Zbigniew, S., Leach, A., Morris, Jeffrey, J., Woodhead, Steven, J., Frederickson, M., Hamlett, C., Woodhead, Andrew, J., Verdonk, Marinus, L., Sore, Hannah, F., Walker, David, W., Blurton, P., Collins, I. & Cheung, Kwai, M., 26 Jun 2008, IPC No. C07D 519/ 00 A I, Patent No. WO2008075109, Priority date 25 Oct 2007, Priority No. US20070982633P

    Research output: Patent

  • SULFONAMIDE DERIVATIVES FOR THERAPEUTIC USE AS FATTY ACID SYNTHASE INHIBITORS

    Butlin, Roger, J., Caulkett, Peter, William, R., Johannesson, P., Knerr, Laurent, D., Leach, A., Newcombe, Nicholas, J., O'Donnell, Charles, J., Pointon, H. & Wood, James, M., 26 Jun 2008, IPC No. C07D 513/ 04 A I, Patent No. WO2008075070, Priority date 5 Apr 2007, Priority No. US20070910232P

    Research output: Patent

  • 2007

    PYRIMIDINE DERIVATIVES

    Kettle, Jason, G., Read, J., Leach, A., Barlaam, Bernard, C., Ducray, R. & Lambert-Van Der Brempt, Christine, M. P., 2 Aug 2007, Patent No. WO2007085833, Priority date 26 Jan 2006, Priority No. US20060762387P

    Research output: Patent