Overcoming the limitations of fragment merging: Rescuing a strained merged fragment series targeting mycobacterium tuberculosis CYP121

Sean A. Hudson, Sachin Surade, Anthony G. Coyne, Kirsty J. Mclean, David Leys, Andrew W. Munro, Chris Abell

    Research output: Contribution to journalArticlepeer-review

    Original languageEnglish
    Pages (from-to)1451-1456
    Number of pages5
    JournalChemMedChem
    Volume8
    Issue number9
    DOIs
    Publication statusPublished - Sept 2013

    Keywords

    • Conformation analysis
    • Cytochromes
    • Drug discovery
    • Fragment-based
    • Tuberculosis

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